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 SUBSTRATES - CYTOCHROME P450 (CYP) ENZYMES DRUG TABLE
CYP1A2  CYP2B6
CYP2C8
CYP2C9
CYP2C19
CYP2D6
CYP2E1
CYP3A4
Genetic
Polymorphisms

    Genetic Polymorphisms
Genetic Polymorphisms
Genetic
Polymorphisms

   
Acetaminophen
Amitriptyline
Asenapine Bendamustine
Caffeine
Chlordiazepoxide
Chlorpromazine
Clopidogrel
Clozapine
Cyclobenzaprine Febuxostat
Flutamide
Imipramine
Leflunomide Mexiletine
Nabumetone
Naproxen
Nortiptyline  Olanzapine Propafenone
Propranolol
Ranitidine
Roflumilast
Riluzole
Tacrine
Theophylline
Tizanidine
Zileuton Zolpidem

Bupropion
Cyclophosphamide
Clopidogrel
Efavirenz
Ifosfamide
Ketamine
Methadone
Sertraline

Amiodarone
Amodiaquine
Benzphetamine Carbamazepine
Cerivastatin
Docetaxel
Everolimus
Febuxostat
Fluvastatin
Isotretinoin
Phenytoin
Pioglitazone
Retinol
Repaglinide
Rosiglitazone
Tolbutamide
Torsemide
Verapamil
Zopiclone

Amitriptyline
Carvedilol
Celecoxib
Chlorpheniramine
Chloramphenicol
Clomipramine
Clopidogrel
Desogstrel
Diclofenac
Dronabinol
Febuxostat
Fluoxetine
Flurbiprofen
Fluvastatin
Formoterol
Glibenclamide
Glimepiride
Glipizide
Hexobarbital
Ibuprofen
Imipramine
Indomethacin
Irbesartan
Irinotecan
Ketamine
Lomoxicam
Losartan
Mefenamic acid
Meloxicam
Mephenytoin
Montelukast
Nateglinide
Omeprazole
Phenylbutazone
Piroxicam
Quetiapine
Rosiglitazone
Sertraline
Sildenafil
Sulfamethoxazole
Sulfinpyrazone
Suprofen
Tamoxifen
Tienilic acid
Tolbutamide

Torsemide
THC
Testosterone
Valdecoxib
Vardenafil
Valsartan
Voriconazole
Warfarin (s)
Zafirlukast
Zileuton

Amitriptyline
Carisoprodol
Cilostazol
Citalopram
Clomipramine
Clopidogrel
Cyclophosphamide
Desipramine
Diazepam
Escitalopram
Esomeprazole
Formoterol
Hexobarbital
Imipramine
Indomethacin
Lacosamide
Lansoprazole
Loratidine
Mephenytoin (s)

Mephenytoin (r)
Mephobarbital (r)
Moclobemide
Nelfinavir
Milutamide
Notripytline
Omeprazole
Pantoprazole
Pentamidine
Phenobarbital
Phenytoin
Progresterone
Proguanil
Propranolol
Rabeprazole
Ranitidine
Sertraline
Teniposide
Thioridazine
Tolbutamide
Voriconazole
Warfarin (r)

Alprenolol
Amitriptyline
Amphetamine 
Aripirazole
Asenpine Atomoxetine
Bifuralol
Bisoprolol
Captopril
Carvedilol
Cevimeline
Chlorpheniramine
Chlorporamzine
Chlorpropamide
Cinacalcet
Clemastine
Clomipramine
Clozapine
Codeine
Cyclobenzaprine
Darifenacin

Debroquine
Desipramine
Dexfenfluramine
Dextromethorphan
Diphenhydramine
Dolasetron
Donepezil
Doxepin
Duloxetine
Encainide
Fenfluramine
Fluphenazine
Fentanyl
Flecainide
Fluoxetine
Fluvoxamine
Formoterol
Galantamine
Guanoxan
Haloperidol
Hydrocodone
Hydroxyzine
Iloperidone
Imipramine
Indoramin
Lidocaine
Maprotiline
Meperidine
Methadone
Methamphetamine
Methoxyamphetamine
Metoclopramide
Metoprolol
Mexiletine
Minaprine
Mirtazapine
Morphine
Nebivolol
Nortriptyline
Olanzapine
Ondansetron
Oxycodone
Paroxetine
Perhexiline
Perphenazine
Propafenone
Propoxyphene
Propranolol
Quetiapine
Quinidine
Ranolazine
Risperidone
Ritonavir
Sertraline
Sparteine
Tamoxifen
Thioridazine
Timolol
Tolterodine
Tramadol
Trazadone
Tripelennamine
Tropisetron
Venlafaxine

Acetaminophen
Disulfiram
Theophylline

Abiraterone
Alfentanil
Alfuzosin
Aliskiren
Almotriptan
Alprazolam
Amitriptyline
Amiodarone
Amlodipine
Amprenavir
Aprepitant
Aripiprazole
Astemizole
Atazanavir
Atorvastatin
Bepridil
Bexarotene
Boceprevir
Bromocriptine
Budesonide
Buprenorphine
Buspirone
Cafergot
Caffeine
Cannabinoids
Carbamazepine
Cerivastatin
Cevimeline
Chlordiazepoxide Cilostazol
Cinacalcet
Citalopram
Clarithromycin
Clindamycin
Clomipramine
Clonazepam
Clopidogrel
Clorazepate
Clozapine
Cocaine
Codeine
Colchicine
Cyclophosphamide
Cyclosporine
Dapsone
Darifenacin
Darunavir
Delavirdine
Desogestrel
Dextromethorphan
Diazepam
Dihdroergotamine
Disopyramide
Diltiazem
Docetaxel
Dofetilide
Dolasetron
Domperidone
Donepezil
Doxorubicin
Dronabinol
Dutasteride
Efavirenz
Eplerenone
Ergotamine
Erlotinib

Erythromycin
Esomeprazole
Eszoplicone
Ethinylestradiol
Ethosuximide
Etonogestrel
Etoposide
Everolimus
Exemestane
Felodipine
Fentanyl
Finasteride
Fexofenadine
Flurazepam Flutamide
Fluticasone
Galantamine
Haloperidol
Hydrocodone
Iloperidone
Imatinib
Imipramine
Indinavir
Irinotecan
Isradipine
Itraconazole
Ketamine
Ketoconazole
Lansoprazole
Letrozole
Lercanidipine
Lidocaine
Loratadine
Lopinavir
Lovastatin
Methadone
Midazolam
Mifepristone
Mirtazapine
Modafinil
Mometasone
Montelukast
Nateglinide
Nelfinavir
Nevirapine
Nicardipine
Nifedipine
Nisoldipine
Nitrendipine
Norethindrone
Ondansetron
Omeprazole
Oxybutynin
Oxycodone
Paclitaxel
Pantoprazole
Pioglitazone
Propafenone Propranolol
Quetiapine
Quinidine
Quinine
Rabeprazole
Ramelteon
Ranitidine
Ranolazine
Repaglinide
Rifampin
Rifaximin
Ritonavir
Rivaroxaban
Rofulmilast
Salmeterol
Saquinavir
Saxagliptin
Sertraline
Sibutramine
Sildenafil
Simvastatin
Sirolimus
Solifenacin
Sorafenib
Sufentanil
Sunitinib
Steroids
Tacrolimus
Tadalafil
Tamoxifen
Telaprevir
Telithromycin
Temazepam
Temsirolimus
THC

Theophylline
Tiagabine
Ticagrelor
Tinidazole
Tipranavir
Tolterodine
Toremifene
Tramadol
Trazadone
Triazolam
Trimetrexate
Valdecoxib
Valproic acid
Vardenafil
Verapamil
Vinblastine
Vincristine
Voriconazole
Warfarin (r)
Zaleplon
Zileuton
Ziprasidone
Zolpidem
Zonisamide


Cytochrome P450 (CYP450) Drug Reference Table - Medication Substrates.